X-Chem delivers excellence, innovation and efficiency at each stage of drug discovery. Since 2012, our medicinal chemists have been named as co-inventors on 24 projects, have filed over 100 patents and published more than 65 scientific papers. Our impressive track record includes 17 compounds reaching IND-enabling toxicology studies and seven compounds progressing to Phase I clinical trials or beyond.

Hit → Lead → Candidate: Click through our proven track record of reliability, efficiency and success.

ION Channels
Target: Sodium Channel Modulator
Therapy Area: Epilepsy
GPCRs
Target: H4 Antagonist
Therapy Area: Inflammation
Transcription Factors
Target: FOXO1 Inhibitor
Therapy Area: Diabetes
Kinases
Target: PINK1 Activator
Therapy Area: Neurodegeneration
Protein Protein Interactions
Target: NLRP3 Inhibitor
Therapy Area: Inflammation
GPCRs
Target: CXCR7 Modulator
Therapy Area: Heart Failure
Protein Protein Interactions
Target: KEAP1 Inhibitor
Therapy Area: Neurodegeneration
GTPASEs
Target: Rac Inhibitor
Therapy Area: Cancer
Epigenetic Regulators
Target: Bromodomain Inhibitor
Therapy Area: Inflammation and Cancer
Epigenetic Regulators
Target: Bromodomain Inhibitor
Therapy Area: Inflammation and Cancer
Epigenetic Regulators
Target: Bromodomain Inhibitor
Therapy Area: Inflammation and Cancer
Epigenetic Regulators
Target: EED (PRC2) Modulator
Therapy Area: Blood Disorder
Epigenetic Regulators
Target: Bromodomain Inhibitor
Therapy Area: Inflammation and Cancer
GPCRs
Target: PAR2 Modulator
Therapy Area: Inflammation
ION Channels
Target: Sodium Channel Modulator
Therapy Area: Epilepsy
Lipids
Target: Ferroptosis Inhibitor
Therapy Area: Neurodegeneration