Scientific Publication Chemical ligation methods for the tagging of DNA-encoded chemical libraries. March 8, 2015
Patents Mitokinin, Inc., USA .; Preparation of purinamines and pyrrolopyrimidinamines, compositions and methods of using the same for treatment of neurodegenerative and mitochondrial disease August 10, 2020
Patents Fulcrum Therapeutics, Inc., USA .; Macrocyclic azolopyridine derivatives as EED and PRC2 modulators and their preparation March 13, 2020
Scientific Publication Asymmetric Synthesis of a Potent CXCR7 Modulator Featuring a Hindered Tertiary Ξ²-Amino Amide Stereocenter August 15, 2018
Scientific Publication Multiple roles of transient receptor potential (TRP) channels in inflammatory conditions and current status of drug development January 2, 2013
Scientific Publication Discovery of a selective c-MET inhibitor with a novel binding mode August 17, 2022
Scientific Publication An integrated approach to fragment-based lead generation: philosophy, strategy and case studies from AstraZeneca’s drug discovery programmes July 15, 2007
Scientific Publication Discovery of Novel, Potent Inhibitors of Hydroxy Acid Oxidase 1 (HAO1) Using DNA-Encoded Chemical Library Screening May 6, 2021
Scientific Publication Novel Nucleic Acid Binding Small Molecules Discovered Using DNA-Encoded Chemistry. May 27, 2019